SCHEMBL8428857

SCHEMBL8428857

COc1ccc(CCNOC(=O)C(C(=O)NCCc2ccc(OC)c(OC)c2)c2ccccc2)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
KMT2A Q03164 5/20 0.55
MEN1 O00255 3/20 0.55
ADRB2 P07550 1/20 0.53
PLAAT3 P53816 1/20 0.53
PLAAT5 Q96KN8 1/20 0.53
PLAAT2 Q9NWW9 1/20 0.53
PLAAT4 Q9UL19 1/20 0.53
MAPT P10636 1/20 0.53
MAPK1 P28482 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
HPGD P15428 1/20 0.52
ALOX12 P18054 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
GAA P10253 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8428854 0.88 ALDH1A1 (0.61) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL742343 0.83 KMT2A (0.71) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL11211724 0.82 ALDH1A1 (0.55) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL6094268 0.82 ALDH1A1 (0.62) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL8098635 0.82 ALDH1A1 (0.62) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL20418416 0.81 ALDH1A1 (0.61) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL11509318 0.81 ALDH1A1 (0.61) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL6376353 0.80 POLB (0.68) ALDH1A1KMT2AMEN1ADRB2PLAAT3
SCHEMBL7442139 0.79 KMT2A (0.66) ALDH1A1KMT2AMEN1MAPTCA12
SCHEMBL8428853 0.79 MEN1 (0.62) ALDH1A1KMT2AMEN1MAPTCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861412-A CARDIOPROTECTIVE AGENTS, CEREBROPROTECTIVE AGENTS, AGENTS FOR TREATING CHRONIC INFLAMMATORY PROCESSES, ANTIPROLIFERATIVE AGENTS AND AS AGENTS FOR TREATING ULCERATIVE COLITIS AND CROHN'S DISEASE BOEHRINGER INGELHEIM KG (DE) 1999-01-19 US disclosed
US-5674878-A ANTIPROLIFERATIVE,-TUMOR AND -CARCINOGENIC AGENTS; ULCERATIVE COLITIS; CROHN*S DISEASE BOEHRINGER INGELHEIM KG (DE) 1997-10-07 US disclosed
US-5643919-A TREATMENT OF CROHN*S DISEASE, ULCERATIVE COLITIS BOEHRINGER INGELHEIM KG (DE) 1997-07-01 US disclosed