SCHEMBL8428876

SCHEMBL8428876

CC(C)CC(=O)N(N)[C@](C(=O)O)(C(=C=O)c1ccccc1)c1cc(NC=NN)cc(C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 2/20 0.35
TACR1 P25103 7/20 0.35
ALDH1A1 P00352 1/20 0.35
RAPGEF3 O95398 3/20 0.33
RAPGEF4 Q8WZA2 2/20 0.33
CTSL P07711 2/20 0.33
TRPA1 O75762 1/20 0.33
CYP1A2 P05177 1/20 0.33
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
TP53 P04637 1/20 0.32
ACP1 P24666 1/20 0.32
PTPN7 P35236 1/20 0.32
PTPN12 Q05209 1/20 0.32
PTPN13 Q12923 1/20 0.32
SSU72 Q9NP77 1/20 0.32
CCR2 P41597 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8429207 0.89 P2RX1 (0.36) P2RX1TACR1ALDH1A1RAPGEF3RAPGEF4
SCHEMBL8429040 0.88 P2RX1 (0.34) P2RX1TACR1ALDH1A1RAPGEF3RAPGEF4
SCHEMBL8431037 0.75 DHODH (0.37) ALDH1A1TP53
SCHEMBL8430960 0.75 MAPT (0.35) ALDH1A1CYP1A2
SCHEMBL8431435 0.74 CA1 (0.32) ALDH1A1TP53
SCHEMBL8431235 0.74 RXFP1 (0.32) CYP1A2
SCHEMBL8429055 0.73 TRPV4 (0.35) CYP1A2
SCHEMBL8521199 0.71 ALDH1A1 (0.36) ALDH1A1
SCHEMBL8432441 0.71 KMT2A (0.32) CYP1A2
SCHEMBL8431423 0.69 DHODH (0.34) ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed