SCHEMBL8428979

SCHEMBL8428979

O=C(CCCCl)N1c2ccccc2Sc2ccccc21

nearest known ligand 0.71

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.70
BCHE P06276 7/20 0.68
ADRB3 P13945 1/20 0.68
HRH2 P25021 1/20 0.68
ADRA1D P25100 1/20 0.68
HTR2A P28223 1/20 0.68
SLC6A4 P31645 1/20 0.68
SLC6A3 Q01959 1/20 0.68
ACHE P22303 4/20 0.63
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
USP2 O75604 1/20 0.54
ALDH1A1 P00352 1/20 0.54
ALOX15 P16050 1/20 0.54
NOX1 Q9Y5S8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11618894 0.90 BCHE (0.67) MAPK1BCHEADRB3HRH2ADRA1D
SCHEMBL8428842 0.89 MEN1 (0.78) MAPK1BCHEADRB3HRH2ADRA1D
SCHEMBL2681239 0.83 BCHE (0.70) MAPK1BCHEADRB3HRH2ADRA1D
SCHEMBL4556566 0.83 MAPK1 (0.68) MAPK1BCHEADRB3HRH2ADRA1D
SCHEMBL8970221 0.81 MAPK1 (0.67) MAPK1BCHEADRB3HRH2ADRA1D
SCHEMBL7982855 0.80 BCHE (0.67) MAPK1BCHEADRB3HRH2ADRA1D
SCHEMBL20272375 0.80 BCHE (0.71) MAPK1BCHEADRB3HRH2ADRA1D
SCHEMBL11171388 0.80 BCHE (0.75) BCHEACHEMEN1KMT2AALDH1A1
SCHEMBL31256024 0.77 NPC1 (0.71) MAPK1MEN1KMT2AALDH1A1
SCHEMBL20272371 0.76 BCHE (0.61) MAPK1BCHEADRB3HRH2ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861394-A COMPOUNDS AS ANTIISCHEMIC AGENTS, TREATMENT OF STROKES, ANTIHEMORRHEGENIC AGENTS, ANTIDEPRESSANTS OR TREATMENT OF SICKKLE CELL ANEMIA BAYER AKTIENGESELLSCHAFT (DE) 1999-01-19 US claimed