SCHEMBL8429186

SCHEMBL8429186

COc1ccccc1C[C@@H](C(=O)Oc1cccc(NC(=N)N)c1)N(NC=O)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.39
ITGB7 P26010 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 3/20 0.34
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
RAB9A P51151 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
PLAU P00749 2/20 0.33
F9 P00740 1/20 0.33
F10 P00742 1/20 0.33
P2RX4 Q99571 1/20 0.33
P2RY14 Q15391 1/20 0.33
MEN1 O00255 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8432434 0.90 PLAU (0.36) SMN1; SMN2MAPTNPC1TP53RAB9A
SCHEMBL8428894 0.89 BACE1 (0.36) ITGA4ITGB7MAPTTP53RAB9A
SCHEMBL8429053 0.89 BACE1 (0.36) ITGA4ITGB7MAPTTP53RAB9A
SCHEMBL8431230 0.82 RAB9A (0.40) NPC1TP53RAB9APLAUKMT2A
SCHEMBL8432438 0.80 RAB9A (0.37) TP53RAB9APLAUALDH1A1PDK1
SCHEMBL8431034 0.79 ALDH1A1 (0.41) SMN1; SMN2MAPTTP53RAB9ANPSR1
SCHEMBL8430957 0.78 PLAU (0.38) TP53RAB9APLAUALDH1A1
SCHEMBL8429153 0.78 SIRT2 (0.37) TP53RAB9APLAUALDH1A1
SCHEMBL8430965 0.78 PDK1 (0.36) TP53RAB9APLAUALDH1A1PDK1
SCHEMBL8430868 0.76 RAB9A (0.41) ITGA4ITGB7MAPTRAB9ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed