SCHEMBL8430223

SCHEMBL8430223

Cc1ccc2c3c(-c4ccc(Cl)cc4)c-3c(Cc3nnn[nH]3)c2c1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.33
GRM2 Q14416 1/20 0.33
FLT1 P17948 1/20 0.32
KDR P35968 1/20 0.32
IKBKB O14920 1/20 0.32
MAP3K14 Q99558 1/20 0.32
TSPO P30536 1/20 0.31
KMT2A Q03164 2/20 0.31
GFER P55789 1/20 0.31
MAP2K4 P45985 4/20 0.31
ALOX12 P18054 1/20 0.31
MAPK1 P28482 3/20 0.31
MAPKAPK3 Q16644 3/20 0.31
MAPK6 Q16659 3/20 0.31
MAPKAPK2 P49137 2/20 0.31
TACR1 P25103 1/20 0.30
MAPKAPK5 Q8IW41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8430246 0.90 MAP2 (0.36) TSPOMAP2K4MAPK1
SCHEMBL8430237 0.86 ESR1 (0.39) KMT2AMAP2K4ALOX12MAPK1
SCHEMBL8430303 0.81 MEN1 (0.40) KMT2AMAPK1
SCHEMBL6505678 0.69 NR1H2 (0.41) KMT2AALOX12
SCHEMBL7484772 0.67 PTGS2 (0.52)
SCHEMBL7484432 0.67 PTGS2 (0.48)
SCHEMBL7482816 0.66 KMT2A (0.31) KMT2A
SCHEMBL7487942 0.66 GPR17 (0.43)
SCHEMBL8430715 0.64 IKBKB (0.32) IKBKBMAP3K14
SCHEMBL17482010 0.64 CHEK1 (0.38) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965619-A ADMINISTERING AN INDENE DERIVATIVE OF GIVEN FORMULA, SUCH AS 1-(2,4,6-TRIMETHOXYBENZYLIDENE)-5-DIMETHYLAMINO-2-METHYL-3-INDENYL ACETIC ACID, TO TREAT PRECANCEROUS LESIONS SUCH AS COLONIC ADENOMATOUS POLYPS; SIDE EFFECT REDUCTION CELL PATHWAYS INC. (US) 1999-10-12 US disclosed