SCHEMBL8430246

SCHEMBL8430246

Clc1ccc(-c2c3c(Cc4nnn[nH]4)c4cc(Cl)ccc4c2-3)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2 P11137 3/20 0.36
CYP19A1 P11511 2/20 0.33
TSPO P30536 1/20 0.33
MAP2K4 P45985 2/20 0.33
EGFR P00533 1/20 0.32
ERBB2 P04626 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
HPGD P15428 1/20 0.31
CYP2C19 P33261 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PTGS2 P35354 2/20 0.31
GPR84 Q9NQS5 2/20 0.31
ROCK2 O75116 1/20 0.30
MAP4K4 O95819 1/20 0.30
LCK P06239 1/20 0.30
CSF1R P07333 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8430237 0.90 ESR1 (0.39) MAP2MAP2K4CYP1A2CYP3A4CYP2C19
SCHEMBL8430223 0.90 DHODH (0.33) TSPOMAP2K4MAPK1
SCHEMBL8430303 0.85 MEN1 (0.40) ALDH1A1HPGDSMN1; SMN2MAPK1
SCHEMBL7487942 0.72 GPR17 (0.43) PTGS2
SCHEMBL7484865 0.69 GPR84 (0.36) GPR84GSK3B
SCHEMBL7479114 0.69 GPR84 (0.36) ALDH1A1GPR84GSK3BDYRK1A
SCHEMBL6505678 0.69 NR1H2 (0.41) KDM4EALDH1A1
SCHEMBL7492466 0.67 GPR17 (0.41) PTGS2
SCHEMBL7487808 0.66 PTGS2 (0.49) PTGS2
SCHEMBL7482841 0.66 PTGS2 (0.47) PTGS2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965619-A ADMINISTERING AN INDENE DERIVATIVE OF GIVEN FORMULA, SUCH AS 1-(2,4,6-TRIMETHOXYBENZYLIDENE)-5-DIMETHYLAMINO-2-METHYL-3-INDENYL ACETIC ACID, TO TREAT PRECANCEROUS LESIONS SUCH AS COLONIC ADENOMATOUS POLYPS; SIDE EFFECT REDUCTION CELL PATHWAYS INC. (US) 1999-10-12 US disclosed