SCHEMBL8431925

SCHEMBL8431925

NCCNC(=O)CCS

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12231859 0.86 HDAC3 (0.42)
SCHEMBL13998028 0.86 HDAC3 (0.46)
SCHEMBL38654455 0.85 ALDH1A1 (0.42)
SCHEMBL12642842 0.83 PAOX (0.53)
SCHEMBL4760493 0.82
SCHEMBL928881 0.82
SCHEMBL636785 0.81
SCHEMBL8436063 0.80
SCHEMBL14198853 0.80 SLC6A5 (0.49)
SCHEMBL13886236 0.80 DNM1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973575-B1 BIOCOMPATIBLE FLUORESCENT METAL OXIDE NANOPARTICLES VISEN MEDICAL INC (US) 2019-07-24 EP disclosed
WO-2016019340-A1 POLYOXAZOLINE ANTIBODY DRUG CONJUGATES SERINA THERAPEUTICS, INC. (US) 2016-02-04 WO disclosed
WO-2011072627-A2 DENDRITIC HIGH-MOLECULAR-WEIGHT POLYMER DRUG CARRIERS AND THEIR CONJUGATES WITH DRUGS ESPECIALLY FOR TREATMENT OF SOLID TUMOURS USTAV MAKROMOLEKULARNI CHEMIE AV CR, V.V.I. (CZ) 2011-06-23 WO disclosed
US-6004531-A LIGANDS FOR RADIOPHARMACEUTICALS; CAPABLE OF CHELATING RADIOMETAL SPECIES AND OF BEING BOUND TO BIOLOGICAL TARGETING MOLECULES NYCOMED AMERSHAM PLC (GB) 1999-12-21 US disclosed
US-5932707-A Thioether-containing metal chelating compounds NYCOMED AMERSHAM PLC (GB) 1999-08-03 US disclosed
WO-1994022816-A1 METAL CHELATING COMPOUNDS AMERSHAM INTERNATIONAL PLC (GB) 1994-10-13 WO disclosed
EP-0618191-A1 Metal chelating compounds AMERSHAM INTERNATIONAL plc (GB) 1994-10-05 EP disclosed