SCHEMBL8432161

SCHEMBL8432161

COc1ccc(C(=O)NCC(=O)NCc2ccccc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.69
RAB9A P51151 4/20 0.69
ALDH1A1 P00352 3/20 0.66
CYP1A2 P05177 1/20 0.66
CYP2D6 P10635 1/20 0.66
CYP2C9 P11712 1/20 0.66
ALOX12 P18054 1/20 0.66
CYP2C19 P33261 1/20 0.66
NPSR1 Q6W5P4 1/20 0.66
POLB P06746 1/20 0.63
CTDSP1 Q9GZU7 1/20 0.63
HPGD P15428 1/20 0.62
TSHR P16473 1/20 0.61
PLA2G1B P04054 1/20 0.60
ATG4B Q9Y4P1 1/20 0.60
MEN1 O00255 1/20 0.59
EPHX2 P34913 1/20 0.59
KMT2A Q03164 1/20 0.59
NR1H4 Q96RI1 1/20 0.59
L3MBTL1 Q9Y468 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2918147 0.90 NPC1 (0.83) NPC1RAB9AALDH1A1CYP1A2CYP2D6
SCHEMBL21773960 0.85 HDAC6 (0.62) RAB9AALDH1A1CTDSP1HPGDMEN1
SCHEMBL2526264 0.84 NPC1 (0.83) NPC1RAB9AALDH1A1CYP1A2CYP2D6
SCHEMBL9416606 0.82 NPC1 (0.82) NPC1RAB9AALDH1A1CYP1A2CYP2D6
SCHEMBL11761142 0.82 NPC1 (0.82) NPC1RAB9AALDH1A1CYP1A2CYP2D6
SCHEMBL1926263 0.82 NPC1 (1.00) NPC1RAB9AALDH1A1CYP1A2CYP2D6
SCHEMBL8213132 0.81 SLC6A9 (0.60) RAB9ACYP1A2CYP2C19HPGDMEN1
SCHEMBL11022457 0.80 FPR2 (0.60) NPC1RAB9AALDH1A1POLBCTDSP1
SCHEMBL5862101 0.80 NPC1 (1.00) NPC1RAB9AALDH1A1CYP2C9CYP2C19
SCHEMBL28497417 0.80 NPC1 (1.00) NPC1RAB9AALDH1A1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0960084-A1 NOVEL SOLID-PHASE SYNTHESIS TECHNIQUES FOR PREPARING MULTIPLE ANALOGOUS COMPOUNDS AXYS PHARMACEUTICALS, INC. (US) 1999-12-01 EP disclosed
WO-1998033751-A1 NOVEL SOLID-PHASE SYNTHESIS TECHNIQUES FOR PREPARING MULTIPLE ANALOGOUS COMPOUNDS AXYS PHARMACEUTICALS, INC. (US) 1998-08-06 WO disclosed