SCHEMBL8434692

SCHEMBL8434692

CC(C)(C)OC(=O)N1CCC[C@H]1CCOc1cccnc1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.52
CHRNA4 P43681 2/20 0.52
CHRNB1 P11230 2/20 0.52
CHRNB4 P30926 2/20 0.52
CHRNA3 P32297 2/20 0.52
CHRNB3 Q05901 2/20 0.52
CHRNA1 P02708 1/20 0.52
CHRNA7 P36544 1/20 0.52
CHEK2 O96017 1/20 0.49
GPR119 Q8TDV5 1/20 0.46
ALOX5AP P20292 1/20 0.44
FEN1 P39748 1/20 0.44
HRH2 P25021 1/20 0.43
HRH1 P35367 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
FKBP1A P62942 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6613800 0.98 CHEK2 (0.52) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL7838155 0.90 CHRNB2 (0.62) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL4143381 0.90 CHRNB2 (0.62) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL7418188 0.90 CHRNB2 (0.62) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL6609250 0.84 CHEK2 (0.56) CHEK2HRH2HRH1KDM4EALDH1A1
SCHEMBL7406714 0.84 CHRNA7 (0.55) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL8440481 0.83 CHRNB1 (0.45) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL8436877 0.83 CHEK2 (0.51) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL611452 0.82 CHRNB2 (0.43) CHRNB2CHRNA4CHRNB1CHRNB4CHRNA3
SCHEMBL4317069 0.79 CHEK2 (0.52) CHEK2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948793-A 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling neurotransmitter release ABBOTT LABORATORIES (US) 1999-09-07 US disclosed
US-5914328-A CONTROL DOPAMINE RELEASE, ACTIVATE CHOLINERGIC CHANNELS ABBOTT LABORATORIES (US) 1999-06-22 US disclosed