SCHEMBL8434724

SCHEMBL8434724

COC(C)OCOc1cc(C(=O)Nc2ccc(C(=O)O)cc2)ccc1C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 11/20 0.44
IKBKB O14920 6/20 0.44
RARB P10826 7/20 0.43
RARG P13631 7/20 0.43
CYP26A1 O43174 3/20 0.43
CYP3A4 P08684 3/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
CYP2C19 P33261 1/20 0.43
PKM P14618 2/20 0.41
PGR P06401 2/20 0.40
NR1I2 O75469 1/20 0.40
LMNA P02545 1/20 0.40
HSPD1 P10809 1/20 0.40
GOT1 P17174 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8424858 0.93 RARA (0.52) RARAIKBKBRARBRARGCYP26A1
SCHEMBL8437029 0.91 RARA (0.41) RARAIKBKBRARBRARGCYP3A4
SCHEMBL8397880 0.90 RARA (0.48) RARAIKBKBRARBRARGCYP3A4
SCHEMBL8396578 0.86 CHEK1 (0.48) MEN1KMT2AALDH1A1MAPK1
SCHEMBL8437023 0.86 RARA (0.41) RARAIKBKBRARBRARGCYP26A1
SCHEMBL8431711 0.85 RARA (0.43) RARAIKBKBRARBRARGCYP3A4
SCHEMBL8434728 0.85 RARA (0.60) RARAIKBKBRARBRARGCYP26A1
SCHEMBL8431940 0.84 CYP3A4 (0.49) RARAIKBKBRARBRARGCYP26A1
SCHEMBL8432347 0.84 HIF1A (0.38) RARAIKBKBRARBCYP2C9PGR
SCHEMBL8435855 0.84 RARA (0.42) RARAIKBKBRARBRARGMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0776881-B1 Bi-aromatic compounds comprising an adamantyl group in para-position, pharmaceutical and cosmetic compositions containing them and their utilization CIRD GALDERMA (FR) 1999-12-08 EP claimed
EP-0776881-B1 Bi-aromatic compounds comprising an adamantyl group in para-position, pharmaceutical and cosmetic compositions containing them and their utilization CIRD GALDERMA (FR) 1999-12-08 EP disclosed
EP-0776881-A1 Bi-aromatic compounds comprising an adamantyl group in para-position, pharmaceutical and cosmetic compositions containing them and their utilization CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (C.I.R.D. GALDERMA) (FR) 1997-06-04 EP disclosed