SCHEMBL8434825

SCHEMBL8434825

COc1ccc2c(c1)C(=O)C(CCCC(=O)O)CC2

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.60
CYP24A1 Q07973 4/20 0.51
CYP26A1 O43174 2/20 0.51
CYP27A1 Q02318 2/20 0.48
METAP1 P53582 1/20 0.47
NQO2 P16083 8/20 0.47
MTNR1A P48039 8/20 0.47
MTNR1B P49286 8/20 0.47
PPARD Q03181 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4623118 0.91 CYP24A1 (0.63) CYP19A1CYP24A1CYP26A1CYP27A1METAP1
SCHEMBL7166421 0.87 CYP24A1 (0.61) CYP19A1CYP24A1CYP26A1CYP27A1METAP1
SCHEMBL7295884 0.85 CYP19A1 (0.65) CYP19A1CYP24A1CYP26A1CYP27A1METAP1
SCHEMBL8028175 0.85 CYP19A1 (0.61) CYP19A1CYP24A1CYP26A1CYP27A1METAP1
SCHEMBL7228543 0.84 CYP19A1 (0.53) CYP19A1CYP24A1CYP26A1NQO2MTNR1A
SCHEMBL4621209 0.83 CYP24A1 (0.65) CYP19A1CYP24A1CYP26A1CYP27A1METAP1
SCHEMBL6645779 0.81 PPARD (0.63) NQO2MTNR1AMTNR1BPPARD
SCHEMBL6645774 0.81 PPARD (0.63) NQO2MTNR1AMTNR1BPPARD
SCHEMBL27599825 0.80 ACHE (0.46) NQO2MTNR1AMTNR1B
SCHEMBL7302984 0.79 CYP19A1 (0.60) CYP19A1CYP24A1CYP26A1CYP27A1METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5945561-A ANTIINFLAMMATORY AGENT, RHEUMATIC DISORDERS, SKIN DISORDERS,ANTISCARRING AGENT BRISTOL-MYERS SQUIBB COMPANY (US) 1999-08-31 US disclosed
WO-1998049136-A1 RETINOID-LIKE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-11-05 WO disclosed