SCHEMBL8435278

SCHEMBL8435278

O=C(O)CCc1cccc(CCc2ccccc2)c1

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 14/20 0.80
KEAP1 Q14145 1/20 0.79
HDAC3 O15379 1/20 0.61
MAPK1 P28482 1/20 0.61
ADRA1A P35348 1/20 0.61
HDAC4 P56524 1/20 0.61
SLC6A3 Q01959 1/20 0.61
HDAC1 Q13547 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
HDAC7 Q8WUI4 1/20 0.61
HDAC2 Q92769 1/20 0.61
HDAC10 Q969S8 1/20 0.61
HDAC11 Q96DB2 1/20 0.61
HDAC8 Q9BY41 1/20 0.61
HDAC6 Q9UBN7 1/20 0.61
HDAC9 Q9UKV0 1/20 0.61
HDAC5 Q9UQL6 1/20 0.61
PTPRB P23467 1/20 0.61
CDC25A P30304 1/20 0.61
CDC25B P30305 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL70271 0.94 KEAP1 (0.74) FFAR1KEAP1HDAC3MAPK1ADRA1A
Hydrochloric Acid SCHEMBL10982620 0.91 KEAP1 (0.71) FFAR1KEAP1HDAC3MAPK1ADRA1A
SCHEMBL12394493 0.89 FFAR1 (1.00) FFAR1KEAP1HDAC3MAPK1ADRA1A
Phenyl Propionic Acid SCHEMBL235064 0.89 KEAP1 (1.00) FFAR1KEAP1HDAC3MAPK1ADRA1A
Phenyl Propionic Acid SCHEMBL29619843 0.89 KEAP1 (1.00) FFAR1KEAP1HDAC3MAPK1ADRA1A
Phenyl Propionic Acid SCHEMBL27523271 0.89 KEAP1 (1.00) FFAR1KEAP1HDAC3MAPK1ADRA1A
Phenyl Propionic Acid SCHEMBL13618844 0.89 KEAP1 (1.00) FFAR1KEAP1HDAC3MAPK1ADRA1A
Phenyl Propionic Acid SCHEMBL3419 0.89 KEAP1 (1.00) FFAR1KEAP1HDAC3MAPK1ADRA1A
Phenyl Propionic Acid SCHEMBL6660445 0.89 KEAP1 (0.68) FFAR1KEAP1HDAC3MAPK1ADRA1A
SCHEMBL29615068 0.88 KEAP1 (0.67) FFAR1KEAP1HDAC3MAPK1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5998433-A THERAPY FOR HYPERLIPIDEMIA; ATHEROSCLEROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-12-07 US disclosed
CN-1160403-A Substd. heterobicyclic alkyl amines and their use as squalene oxide cyclase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-09-24 CN disclosed
EP-0785939-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS Takeda Chemical Industries, Ltd. (JP) 1997-07-30 EP disclosed
WO-1996011201-A1 SUBSTITUTED HETEROBICYCLIC ALKYL AMINES AND THEIR USE AS SQUALENE OXIDE CYCLASE INHIBITORS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-04-18 WO disclosed