SCHEMBL8435340

SCHEMBL8435340

CCC(=O)N(c1ccncc1)c1csc2cnccc12

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
RPS6KB1 P23443 1/20 0.33
CDK2 P24941 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
GSK3B P49841 1/20 0.33
RPS6KA3 P51812 1/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 3/20 0.33
KDM4E B2RXH2 3/20 0.33
CDC7 O00311 3/20 0.33
DBF4 Q9UBU7 3/20 0.33
HSD17B10 Q99714 2/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
CASP1 P29466 1/20 0.33
HTT P42858 1/20 0.33
CASP7 P55210 1/20 0.33
NCOA1 Q15788 1/20 0.33
RCE1 Q9Y256 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8436325 0.90 CYP2A6 (0.39) LMNASMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL7342232 0.87 GAA (0.38) SMN1; SMN2ALDH1A1HPGDKDM4EGAA
SCHEMBL8438852 0.85 CDC7 (0.36) LMNAGSK3BRPS6KA3ALDH1A1HPGD
SCHEMBL8436069 0.78 TRPM8 (0.35) LMNASMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL9004605 0.78 IRAK4 (0.33) LMNASMN1; SMN2ALDH1A1HPGDKDM4E
SCHEMBL8435887 0.77 LATS1 (0.38) GSK3BLATS1LATS2BRAFCYP2A6
SCHEMBL8440253 0.75 CHRM5 (0.38) SMN1; SMN2GSK3BLATS1LATS2BRAF
SCHEMBL8442574 0.75 CYP2A6 (0.41) LMNASMN1; SMN2GSK3BRPS6KA3ALDH1A1
SCHEMBL8436369 0.75 SLC6A2 (0.37) LATS1LATS2BRAFCYP2A6
SCHEMBL7335255 0.74 CYP2A6 (0.38) SMN1; SMN2ALDH1A1HPGDKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856335-A GLYCINE PARTIAL AGONISTS. HOECHST MARION ROUSSEL, INC. (US) 1999-01-05 US disclosed
US-5519032-A ANTIDEPRESSANTS, ANXIOLYTICS, ANTIEMETICS, ANTIPSYCHOTIC HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
EP-0581106-A1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-02-02 EP disclosed
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed