SCHEMBL8438852

SCHEMBL8438852

CC(=O)N(c1ccncc1)c1csc2cnccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.36
PLK4 O00444 1/20 0.36
DAPK3 O43293 1/20 0.36
ROCK2 O75116 1/20 0.36
CHEK2 O96017 1/20 0.36
PIM1 P11309 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
GSK3A P49840 1/20 0.36
GSK3B P49841 1/20 0.36
RPS6KA3 P51812 1/20 0.36
PRKX P51817 1/20 0.36
PLK1 P53350 1/20 0.36
CSNK1G2 P78368 1/20 0.36
PRKCZ Q05513 1/20 0.36
ROCK1 Q13464 1/20 0.36
PRKG1 Q13976 1/20 0.36
CDC42BPA Q5VT25 1/20 0.36
AURKB Q96GD4 1/20 0.36
PLK3 Q9H4B4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8442574 0.89 CYP2A6 (0.41) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8435340 0.85 LMNA (0.34) CDC7GSK3BRPS6KA3KDM4EALDH1A1
SCHEMBL8440253 0.78 CHRM5 (0.38) GSK3BCYP2A6BRAFMAP3K7TAB1
SCHEMBL8442576 0.76 NSD2 (0.36) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8439945 0.76 LMNA (0.34) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8436325 0.75 CYP2A6 (0.39) CDC7ROCK2KDM4EALDH1A1HPGD
SCHEMBL8435887 0.74 LATS1 (0.38) GSK3BCYP2A6BRAFMAP3K7TAB1
SCHEMBL8436369 0.72 SLC6A2 (0.37) CYP2A6BRAFMAP3K7TAB1LATS1
SCHEMBL7342232 0.72 GAA (0.38) KDM4EALDH1A1GAAHPGDCYP2A6
SCHEMBL15573652 0.71 CYP2A6 (0.45) DAPK3PIM1KDRGSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856335-A GLYCINE PARTIAL AGONISTS. HOECHST MARION ROUSSEL, INC. (US) 1999-01-05 US disclosed
US-5519032-A ANTIDEPRESSANTS, ANXIOLYTICS, ANTIEMETICS, ANTIPSYCHOTIC HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
EP-0581106-A1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-02-02 EP disclosed
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed