SCHEMBL8435856

SCHEMBL8435856

O=C(O)C1CCN(S(=O)(=O)c2ccc(OCc3cnc(Cl)s3)cc2)C(C(=O)NO)C1

nearest known ligand 0.58

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 20/20 0.58
MMP1 P03956 17/20 0.58
MMP13 P45452 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431603 0.88 ADAM17 (0.56) ADAM17MMP1MMP13
SCHEMBL8433179 0.82 ADAM17 (0.68) ADAM17MMP1MMP13
SCHEMBL7220235 0.80 MMP1 (0.83) ADAM17MMP1MMP13
SCHEMBL7214512 0.80 MMP1 (0.83) ADAM17MMP1MMP13
SCHEMBL8521842 0.80 ADAM17 (0.58) ADAM17MMP1MMP13
SCHEMBL5760044 0.80 ADAM17 (0.49) ADAM17MMP1MMP13
SCHEMBL8431700 0.79 ADAM17 (0.56) ADAM17MMP1MMP13
SCHEMBL8432178 0.77 ADAM17 (0.58) ADAM17MMP1MMP13
SCHEMBL8573731 0.76 ADAM17 (0.51) ADAM17MMP1MMP13
SCHEMBL8573736 0.76 ADAM17 (0.51) ADAM17MMP1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0960098-A1 ARYLSULFONYL HYDROXAMIC ACID DERIVATIVES PFIZER INC. (US) 1999-12-01 EP disclosed
WO-1998034918-A1 ARYLSULFONYL HYDROXAMIC ACID DERIVATIVES PFIZER INC. (US) 1998-08-13 WO disclosed