SCHEMBL8436255

SCHEMBL8436255

[CH2]C(=O)NCC(CC)CC

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.36
USP2 O75604 1/20 0.36
HTT P42858 2/20 0.33
GLA P06280 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
LMNA P02545 2/20 0.30
POLB P06746 1/20 0.30
MAPK1 P28482 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP3A4 P08684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8350700 0.83 TSHR (0.55) TSHRHTTGLAL3MBTL1LMNA
SCHEMBL8437414 0.78
SCHEMBL3274384 0.77 TSHR (0.37) TSHRUSP2HTTGLAL3MBTL1
SCHEMBL8436259 0.77 MAPK1 (0.40) TSHRUSP2HTTCYP2D6CYP2C19
SCHEMBL3274387 0.77 CYP2D6 (0.56) TSHRUSP2HTTGLAL3MBTL1
SCHEMBL8437855 0.76 TSHR (0.33) TSHRUSP2HTTGLAL3MBTL1
SCHEMBL17624747 0.75 KMT2A (0.48) TSHRUSP2HTTGLAL3MBTL1
SCHEMBL9749983 0.75 BCAT2 (0.39) TSHRUSP2HTTGLAL3MBTL1
SCHEMBL17183684 0.75 TSHR (0.50) TSHRUSP2HTTGLAL3MBTL1
SCHEMBL459003 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088120-A inhibitors of transglutaminase 策迪拉有限公司 2019-08-02 CN disclosed
EP-0777658-B1 SUBSTITUTED TRIAZOLINONES AS PLANT PROTECTIVE AGENTS BASF AG (DE) 1999-12-15 EP disclosed
US-5885934-A HERBICIDES OR FOR THE DESICCATION/DEFOLIATION OF PLANTS BASF AKTIENGESELLSCHAFT (DE) 1999-03-23 US disclosed
EP-0777658-A1 SUBSTITUTED TRIAZOLINONES AS PLANT PROTECTIVE AGENTS BASF AKTIENGESELLSCHAFT (DE) 1997-06-11 EP disclosed
WO-1996005179-A1 SUBSTITUTED TRIAZOLINONES AS PLANT PROTECTIVE AGENTS BASF AKTIENGESELLSCHAFT (DE) 1996-02-22 WO disclosed