SCHEMBL8436760

SCHEMBL8436760

CCCCc1nc(Br)c(Br)[nH]1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MAPK1 P28482 1/20 0.46
PARP1 P09874 1/20 0.40
GPR84 Q9NQS5 5/20 0.39
GSK3B P49841 1/20 0.37
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
PI4KA P42356 1/20 0.36
PI4K2B Q8TCG2 1/20 0.36
PI4K2A Q9BTU6 1/20 0.36
PI4KB Q9UBF8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11360102 0.82 ALDH1A1 (0.44) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL9083256 0.77 ALDH1A1 (0.41) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL27431902 0.77 ALDH1A1 (0.41) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL9122617 0.77 ALDH1A1 (0.41) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL1257638 0.76 ALDH1A1 (0.40) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL9123535 0.76 PARP1 (0.42) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL28455056 0.75 ATM (0.49) ALDH1A1MAPK1GPR84PKMHPGD
SCHEMBL9584829 0.73 GPR84 (0.39) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL8434384 0.73 KDM4E (0.40) ALDH1A1MAPK1PARP1GPR84GSK3B
SCHEMBL9592380 0.72 GPR84 (0.38) ALDH1A1MAPK1PARP1GPR84GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102596937-A Compounds and compositions as protein kinase inhibitors NOVARTIS AG 2012-07-18 CN disclosed
US-5929249-A ANGIOTENSIN II RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-07-27 US disclosed
US-5728842-A ANGIOTENSIN II RECEPTOR ANTAGONIST SMITHKLINE BEECHAM CORPORATION (US) 1998-03-17 US disclosed
EP-0653937-A4 CHEMICAL COMPOUNDS. SMITHKLINE BEECHAM CORP (US) 1996-07-31 EP disclosed
EP-0653937-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1995-05-24 EP disclosed
WO-1994000120-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-01-06 WO disclosed
US-5208235-A Phosphonic or phosphinic acid derivatives as inhibitors of angiotnesin II for cardiovascular disorders and hypotensives E. R. SQUIBB & SONS, INC. (US) 1993-05-04 US disclosed