SCHEMBL8437249

SCHEMBL8437249

COc1ccn(-c2ccc(Cl)c(Cl)c2)n1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 18/20 0.56
KCNH2 Q12809 1/20 0.48
NOTUM Q6P988 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7923053 0.81 SIGMAR1 (0.49) SIGMAR1NOTUM
SCHEMBL16202039 0.78 ALDH1A1 (0.40) SIGMAR1NOTUM
SCHEMBL2615992 0.77 NOTUM (0.51) SIGMAR1NOTUM
SCHEMBL731151 0.77 SIGMAR1 (0.67) SIGMAR1KCNH2
SCHEMBL466979 0.76 SIGMAR1 (0.88) SIGMAR1KCNH2
SCHEMBL27781400 0.75 ABCB11 (0.50)
SCHEMBL28783897 0.75 ALDH1A1 (0.50) NOTUM
Hydrochloric Acid SCHEMBL1903312 0.75 SIGMAR1 (0.86) SIGMAR1KCNH2
SCHEMBL28020284 0.75 NOTUM (0.57) NOTUM
SCHEMBL24891467 0.74 SIGMAR1 (0.46) SIGMAR1KCNH2NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1829873-A1 Pyrrazole derivatives as sigma receptors antagonists LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2007-09-05 EP disclosed