SCHEMBL8438748

SCHEMBL8438748

COc1ccc(OC)c(C#Cc2ccc3nc(C)ncc3c2)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.45
EGFR P00533 1/20 0.40
HPGDS O60760 1/20 0.39
NQO1 P15559 1/20 0.39
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
HAO1 Q9UJM8 1/20 0.36
GRM5 P41594 2/20 0.36
AAK1 Q2M2I8 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7796162 0.82 EGFR (0.63) DHFREGFRHPGDSNQO1PDGFRB
SCHEMBL1161417 0.79 EGFR (0.59) EGFRNQO1PDGFRBPDGFRAMAPT
SCHEMBL8434822 0.76 PDGFRB (0.42) DHFREGFRPDGFRBPDGFRAMAPT
SCHEMBL27878442 0.75 AR (0.49) DHFRHAO1AAK1MAPTHTT
SCHEMBL7803054 0.75 DHFR (0.42) DHFREGFRMAPTHTT
SCHEMBL7796228 0.72 CSF1R (0.42) DHFREGFRPDGFRBPDGFRAHAO1
SCHEMBL27878604 0.71 APP (0.66) DHFRMAPT
SCHEMBL12361591 0.70 EGFR (0.59) EGFRHPGDSPDGFRBPDGFRA
SCHEMBL7804802 0.70 MTNR1A (0.44) DHFREGFRMAPT
SCHEMBL7803061 0.70 IP6K1 (0.58) DHFRHAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990116-A USE IN PREVENTION OR TREATMENT OF INFLAMMATORY AND PROLIFERATIVE SKIN DISEASES AND CANCER; COMPOUNDS SUCH AS 6-(2-(2,5-DIMETHOXYPHENYL)ETHYL)-4-ETHYL-QUINAZOLINE NOVARTIS AG (CH) 1999-11-23 US disclosed