SCHEMBL8439554

SCHEMBL8439554

O=C(O)c1cc(C(=O)O)cc(-c2ccoc2C(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.37
DHODH Q02127 3/20 0.36
TTR P02766 3/20 0.36
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
PTGER1 P34995 1/20 0.34
XDH P47989 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
AURKA O14965 1/20 0.33
TPX2 Q9ULW0 1/20 0.33
HCAR1 Q9BXC0 1/20 0.33
DAO P14920 2/20 0.33
KMO O15229 1/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8443666 0.89 KDM4E (0.39) CA12CA1CA2CA7CA9
SCHEMBL8444445 0.73 CHRM2 (0.51) CA12CA1CA2CA9
SCHEMBL8441952 0.72 KEAP1 (0.38) KEAP1DHODHXDHSLC22A12DAO
SCHEMBL8805333 0.71 HTR2B (0.42)
SCHEMBL8443923 0.68 DHODH (0.36) DHODHTTRPTGER1DAOKMO
SCHEMBL15521796 0.68 CA12 (0.48) DHODHTTRCA12CA1CA2
SCHEMBL8442873 0.67 KEAP1 (0.43) KEAP1DHODHTTRXDHSLC22A12
SCHEMBL29908924 0.67 DHODH (0.57) DHODHTTRPTGER1DAOKMO
SCHEMBL24526667 0.66 PTGER1 (0.43) KEAP1PTGER1HCAR1DAOALDH1A1
SCHEMBL8444491 0.66 TNKS (0.44) DHODHTTRCA1CA2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968985-A INHIBITORS OF SODIUM ION/HYDROGEN ION EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-19 US disclosed
EP-0773927-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-21 EP disclosed
WO-1996004241-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-15 WO disclosed