SCHEMBL8442873

SCHEMBL8442873

O=C(O)c1cc(C(=O)O)cc(-c2cccc3occc23)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.43
DHODH Q02127 4/20 0.40
KMO O15229 1/20 0.39
DAO P14920 1/20 0.38
XDH P47989 1/20 0.38
SLC22A12 Q96S37 1/20 0.38
FTO Q9C0B1 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
TTR P02766 1/20 0.37
BCHE P06276 1/20 0.37
POLB P06746 1/20 0.37
HSP90AA1 P07900 1/20 0.37
HSP90AB1 P08238 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8802708 0.89 KEAP1 (0.53) KEAP1KMOTDP1KDM4EALDH1A1
SCHEMBL8444450 0.82 TNKS (0.40) MEN1KMT2ALMNAMAPTTHRB
Isophthalic Acid SCHEMBL27753681 0.76 PTPN1 (0.50) KEAP1KMOMEN1KMT2AKDM4E
SCHEMBL10578274 0.76 XDH (0.44) KEAP1DHODHKMODAOXDH
SCHEMBL2143620 0.76 MAOB (0.45) FTOMEN1KMT2AKDM4EALDH1A1
SCHEMBL8442957 0.76 CHRM2 (0.49) SMN1; SMN2
SCHEMBL16488681 0.74 DHODH (0.53) DHODHKMODAOTDP1MEN1
SCHEMBL29908924 0.73 DHODH (0.57) DHODHKMODAOKMT2ATTR
SCHEMBL8440725 0.73 CYP4F2 (0.41) MEN1KMT2AKDM4EALDH1A1LMNA
SCHEMBL29908910 0.72 DHODH (0.55) DHODHKMODAOKMT2ATTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968985-A INHIBITORS OF SODIUM ION/HYDROGEN ION EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-19 US disclosed
EP-0773927-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-21 EP disclosed
WO-1996004241-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-15 WO disclosed