SCHEMBL8440389

SCHEMBL8440389

CCN(c1ccncc1)c1csc2ccncc12

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.40
LATS1 O95835 6/20 0.35
LATS2 Q9NRM7 5/20 0.35
CHRM5 P08912 1/20 0.32
CHKA P35790 1/20 0.32
KDM4C Q9H3R0 1/20 0.31
HTR6 P50406 1/20 0.30
SLC6A2 P23975 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8438931 0.89 CYP2A6 (0.41) CYP2A6LATS1LATS2KDM4CHTR6
SCHEMBL8435887 0.88 LATS1 (0.38) CYP2A6LATS1LATS2CHRM5CHKA
SCHEMBL8440769 0.86 LATS1 (0.38) CYP2A6LATS1LATS2HTR6SLC6A2
SCHEMBL8056316 0.85 SLC6A2 (0.38) CYP2A6SLC6A2
Hydrochloric Acid SCHEMBL8039091 0.84 ALDH1A1 (0.40) CYP2A6SLC6A2
SCHEMBL8440409 0.80 CYP2A6 (0.43) CYP2A6LATS1LATS2CHRM5CHKA
SCHEMBL8049764 0.78 MAPK14 (0.33) LATS1LATS2HTR6
SCHEMBL8050470 0.78 ROCK1 (0.37) CYP2A6CHKASLC6A2
SCHEMBL8436369 0.77 SLC6A2 (0.37) CYP2A6LATS1LATS2KDM4CSLC6A2
Hydrochloric Acid SCHEMBL8050473 0.77 MAPK14 (0.33) LATS1LATS2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856335-A GLYCINE PARTIAL AGONISTS. HOECHST MARION ROUSSEL, INC. (US) 1999-01-05 US disclosed
US-5519032-A ANTIDEPRESSANTS, ANXIOLYTICS, ANTIEMETICS, ANTIPSYCHOTIC HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
EP-0581106-A1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-02-02 EP disclosed
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed