SCHEMBL8440769

SCHEMBL8440769

CCCCN(c1ccncc1)c1csc2ccncc12

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LATS1 O95835 4/20 0.38
LATS2 Q9NRM7 4/20 0.38
CYP2A6 P11509 1/20 0.37
SLC6A2 P23975 2/20 0.34
MAPT P10636 2/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTT P42858 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
HTR6 P50406 1/20 0.30
ATP4A P20648 1/20 0.30
ATP4B P51164 1/20 0.30
NR1H2 P55055 1/20 0.30
NR1H3 Q13133 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8438931 0.92 CYP2A6 (0.41) LATS1LATS2CYP2A6SLC6A2HTR6
SCHEMBL8438770 0.90 LATS1 (0.40) LATS1LATS2SLC6A2MAPTMAPK1
SCHEMBL8038900 0.87 SLC6A2 (0.41) LATS1LATS2CYP2A6SLC6A2MAPT
SCHEMBL8440389 0.86 CYP2A6 (0.40) LATS1LATS2CYP2A6SLC6A2HTR6
Hydrochloric Acid SCHEMBL8039092 0.86 SLC6A2 (0.40) CYP2A6SLC6A2MAPTMAPK1NPSR1
SCHEMBL8436369 0.81 SLC6A2 (0.37) LATS1LATS2CYP2A6SLC6A2
SCHEMBL8050077 0.80 MAPT (0.33) LATS1LATS2SLC6A2MAPTMAPK1
SCHEMBL8039432 0.80 SLC6A2 (0.37) LATS1LATS2CYP2A6SLC6A2MAPT
Hydrochloric Acid SCHEMBL9425165 0.79 SLC6A2 (0.37) LATS1LATS2CYP2A6SLC6A2MAPT
Hydrochloric Acid SCHEMBL8056275 0.79 MAPT (0.33) LATS1LATS2SLC6A2MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856335-A GLYCINE PARTIAL AGONISTS. HOECHST MARION ROUSSEL, INC. (US) 1999-01-05 US disclosed
US-5519032-A ANTIDEPRESSANTS, ANXIOLYTICS, ANTIEMETICS, ANTIPSYCHOTIC HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
EP-0581106-A1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-02-02 EP disclosed
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed