SCHEMBL8440455

SCHEMBL8440455

COC(=O)c1cccc(-c2c(C)oc3ccccc23)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 1/20 0.50
CYP2C19 P33261 2/20 0.47
HIF1A Q16665 1/20 0.46
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
ERN1 O75460 2/20 0.43
TP53 P04637 1/20 0.43
NEK1 Q96PY6 1/20 0.43
PDE5A O76074 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8444471 0.86 TNKS (0.49) TNKSCYP2C19HIF1AKDM4ENPC1
SCHEMBL8442687 0.85 CYP2C19 (0.50) TNKSCYP2C19KDM4EMEN1KMT2A
SCHEMBL8443281 0.84 ERN1 (0.49) TNKSHIF1AKDM4ENPC1RAB9A
SCHEMBL8442828 0.83 TNKS (0.46) TNKSHIF1AKDM4ENPC1RAB9A
SCHEMBL8802437 0.79 CYP2C19 (0.43) CYP2C19KDM4ENPC1RAB9AMEN1
SCHEMBL8802443 0.79 HTR2B (0.56) CYP2C19
SCHEMBL12754449 0.77 GPR119 (0.53) TNKSHIF1AKDM4ENPC1RAB9A
SCHEMBL13986661 0.76 ALOX5 (0.52) TNKSHIF1ANPC1RAB9AGABRG2
SCHEMBL8444433 0.76 CYP2C19 (0.40) CYP2C19KDM4ENPC1RAB9AMEN1
SCHEMBL29129510 0.75 MEN1 (0.51) TNKSCYP2C19KDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968985-A INHIBITORS OF SODIUM ION/HYDROGEN ION EXCHANGE IN CELLS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-19 US disclosed
EP-0773927-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-05-21 EP disclosed
WO-1996004241-A2 BENZOYLGUANIDINE DERIVATIVES AS MEDICAMENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-02-15 WO disclosed