SCHEMBL8302305

SCHEMBL8302305

O=C1Cc2cc(C(=O)CN3CCC(CCC4CCCCC4)CC3)ccc2N1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.52
HTR1A P08908 1/20 0.48
DRD2 P14416 1/20 0.48
HTR2A P28223 1/20 0.48
HTR2C P28335 1/20 0.48
HTR7 P34969 1/20 0.48
DRD3 P35462 1/20 0.48
HTR2B P41595 1/20 0.48
SMYD3 Q9H7B4 10/20 0.47
ACHE P22303 5/20 0.45
EPHX2 P34913 2/20 0.45
HTR4 Q13639 2/20 0.45
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8440778 0.90 GRIN2B (0.53) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL8439771 0.86 GRIN2B (0.52) GRIN2BHTR1AHTR2AHTR7DRD3
SCHEMBL7564279 0.86 GRIN2B (0.57) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL5843055 0.85 GRIN2B (0.58) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL9825056 0.80 GRIN2B (0.56) GRIN2BHTR1ADRD2HTR2AHTR2C
Hydrochloric Acid SCHEMBL9825181 0.79 GRIN2B (0.55) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL7210683 0.79 GRIN2B (0.55) GRIN2BHTR1ADRD2HTR2AHTR2C
SCHEMBL8300540 0.78 HTR1A (0.56) HTR1ADRD2HTR2AACHEEPHX2
SCHEMBL8301786 0.77 HTR1A (0.53) GRIN2BHTR1ADRD2HTR2ASMYD3
SCHEMBL9825127 0.76 GRIN2B (0.66) GRIN2BHTR1ADRD2HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848707-B1 4-(CYCLOALKYL)PIPERIDINES AND 4-(CYCLOALKYLALKYL)-PIPERIDINES DERIVATIVES, PREPARATION THEREOF AND THERAPEUTICAL APPLICATIONS THEREOF SYNTHELABO (FR) 1999-08-04 EP disclosed