SCHEMBL8443531

SCHEMBL8443531

Bc1ccc(C(=O)NCCN(C)C)c(O)c1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
CYP1A2 P05177 1/20 0.50
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 2/20 0.49
HSD17B10 Q99714 1/20 0.46
AOX1 Q06278 1/20 0.45
APP P05067 3/20 0.44
RAD52 P43351 2/20 0.44
MAPK1 P28482 1/20 0.43
HPGD P15428 1/20 0.43
ALOX12 P18054 1/20 0.43
HTR2C P28335 1/20 0.43
UHRF1 Q96T88 1/20 0.42
CHEK1 O14757 1/20 0.42
USP2 O75604 1/20 0.42
MCHR1 Q99705 1/20 0.41
ACKR3 P25106 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2823242 0.82 CYP1A2 (0.68) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E
SCHEMBL21046542 0.81 HTT (0.66) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E
SCHEMBL8639778 0.78 NAAA (0.60) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E
SCHEMBL11216405 0.77 KDM4E (0.68) HTTSMN1; SMN2ALDH1A1KDM4EHSD17B10
SCHEMBL19418228 0.76 ALDH1A1 (0.63) HTTSMN1; SMN2ALDH1A1KDM4EHSD17B10
SCHEMBL2848982 0.74 HTT (0.48) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E
SCHEMBL22023523 0.73 HTT (0.54) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E
SCHEMBL16523438 0.73 SMN1; SMN2 (1.00) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E
SCHEMBL30231342 0.72 ACKR3 (0.69) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E
SCHEMBL24163465 0.71 HTT (0.48) HTTSMN1; SMN2CYP1A2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed