SCHEMBL8444030

SCHEMBL8444030

CCn1ncc2c(NCc3cccnc3)c3ccccc3nc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.50
KMT2A Q03164 7/20 0.50
KDM4E B2RXH2 5/20 0.50
GAA P10253 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
POLB P06746 2/20 0.49
RAD52 P43351 1/20 0.49
CYP1A2 P05177 8/20 0.48
CYP3A4 P08684 8/20 0.48
CYP2D6 P10635 8/20 0.48
CYP2C19 P33261 8/20 0.48
PDE5A O76074 3/20 0.48
CYP2C9 P11712 2/20 0.48
TSHR P16473 7/20 0.47
HSD17B10 Q99714 7/20 0.47
MAPK1 P28482 3/20 0.47
CLK4 Q9HAZ1 3/20 0.47
PDE9A O76083 1/20 0.47
MAPT P10636 6/20 0.47
ALOX15 P16050 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7028354 0.91 KMT2A (0.60) ALDH1A1KMT2AKDM4EPOLBRAD52
SCHEMBL7418635 0.89 POLB (0.51) ALDH1A1KMT2AKDM4EL3MBTL1POLB
SCHEMBL7423097 0.83 POLB (0.48) KMT2APOLBRAD52PDE5APDE9A
SCHEMBL7420540 0.83 POLB (0.50) KMT2APOLBRAD52PDE5APDE9A
SCHEMBL7420650 0.82 PDE5A (0.50) ALDH1A1KMT2AKDM4EPOLBRAD52
SCHEMBL13692589 0.82 KMT2A (0.73) ALDH1A1KMT2AKDM4EGAAL3MBTL1
SCHEMBL7425050 0.81 ALDH1A1 (0.47) ALDH1A1KMT2AKDM4EGAAPOLB
SCHEMBL7416586 0.81 EGFR (0.52) ALDH1A1KMT2AGAAPOLBRAD52
SCHEMBL7418464 0.81 APP (0.53) ALDH1A1KMT2AGAAPOLBRAD52
SCHEMBL7418050 0.81 BCHE (0.50) ALDH1A1KMT2AKDM4EGAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6008226-A AN ENZYME INHIBITOR OF C-GMP-PHOSPHODIESTERASE FOR TREATING HEART FAILURE, HYPERTENSION, REVERSING OR REDUCING NITRATE-INDUCED TOLERANCE AND ANGINA PECTORIS, CONGESTIVE HEART DISEASE AND MYOCARDIAL INFARCTION SANOFI-SYNTHELABO (FR) 1999-12-28 US disclosed