SCHEMBL8446366

SCHEMBL8446366

COC(=O)c1ccc(O)c(B(O)O)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.67
CA2 P00918 5/20 0.67
CA12 O43570 4/20 0.67
CA7 P43166 4/20 0.67
CA9 Q16790 4/20 0.67
CA14 Q9ULX7 4/20 0.67
XDH P47989 2/20 0.67
KDM4E B2RXH2 4/20 0.59
ALDH1A1 P00352 3/20 0.59
HPGD P15428 3/20 0.59
HSD17B10 Q99714 3/20 0.59
MAPT P10636 3/20 0.59
LMNA P02545 2/20 0.59
TP53 P04637 2/20 0.59
ALOX15 P16050 2/20 0.59
ALOX12 P18054 2/20 0.59
MEN1 O00255 1/20 0.59
HTT P42858 1/20 0.59
KMT2A Q03164 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18713916 0.85 CA1 (0.67) CA1CA2CA12CA7CA9
SCHEMBL29587663 0.81 TDP1 (0.52) CA1CA2CA12CA7CA9
SCHEMBL2417938 0.81 TDP1 (0.52) CA1CA2CA12CA7CA9
SCHEMBL29952679 0.81 CA12 (0.70) CA1CA2CA12CA7CA9
Methyl Protocatechuate SCHEMBL29360855 0.80 CA1 (1.00) CA1CA2CA12CA7CA9
Methyl Protocatechuate SCHEMBL38624 0.80 CA1 (1.00) CA1CA2CA12CA7CA9
SCHEMBL559758 0.80 ALDH1A1 (0.57) CA1CA2CA12CA7CA9
SCHEMBL701513 0.80 CA1 (0.50) CA1CA2CA12CA7CA9
SCHEMBL30740888 0.80 MAPT (0.60) CA1CA2CA12CA7CA9
SCHEMBL29626852 0.80 CA1 (0.50) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
WO-2010069504-A1 (3-OXO)PYRIDIN-4-YLUREA DERIVATIVES AS PDE4 INHIBITORS ALMIRALL, S.A. (ES) 2010-06-24 WO disclosed
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed