SCHEMBL8448176

SCHEMBL8448176

O=Cc1cc([N+](=O)[O-])c(Br)s1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.42
ALDH5A1 P51649 1/20 0.41
ABAT P80404 1/20 0.41
VCAM1 P19320 1/20 0.41
ALDH1A1 P00352 5/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 2/20 0.38
MAPT P10636 3/20 0.38
ALDH1A3 P47895 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
XDH P47989 1/20 0.37
GPR35 Q9HC97 1/20 0.36
KDM4E B2RXH2 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
HSP90AA1 P07900 1/20 0.36
RECQL P46063 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10745204 0.81 ERN1 (0.37) ERN1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL11269447 0.78 MAPT (0.44) ALDH1A1CYP1A2MAPTTDP1GPR35
SCHEMBL2681533 0.77 VCAM1 (0.44) ERN1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL1187281 0.77 PSMB8 (0.42) ERN1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL12963014 0.77 ALDH1A1 (0.37) ERN1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL2680731 0.75 CYP3A4 (0.39) ERN1ALDH1A1CYP1A2CYP2C19MAPT
SCHEMBL947371 0.74 ERN1 (0.36) ERN1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL10742175 0.73 ALDH1A1 (0.40) ERN1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL11829469 0.73 MAPT (0.35) ERN1ALDH5A1ABATVCAM1ALDH1A1
SCHEMBL11817923 0.73 CYP2A6 (0.41) ERN1ALDH5A1ABATVCAM1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5942387-A Combinatorial process for preparing substituted thiophene libraries ELI LILLY AND COMPANY (US) 1999-08-24 US disclosed
WO-1998008839-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED THIOPHENE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed
US-4659735-A Benzofuranyl (thienyl) propenyl derivatives useful as rodenticides HOFFMANN-LA ROCHE INC. (US) 1987-04-21 US disclosed
US-4649154-A AGRICULTURE DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1987-03-10 US disclosed
US-4451660-A AGRICULTURE, HORTICULTURE DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1984-05-29 US disclosed
EP-0031173-B1 NEW NITROTHIOPHENES, METHOD OF PREPARING THE NEW COMPOUNDS, AS WELL AS FUNGICIDAL AND/OR BACTERICIDAL COMPOSITIONS ON THE BASIS OF THE NEW COMPOUNDS DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1983-09-14 EP disclosed
EP-0031173-A1 New nitrothiophenes, method of preparing the new compounds, as well as fungicidal and/or bactericidal compositions on the basis of the new compounds DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1981-07-01 EP disclosed