SCHEMBL845083

SCHEMBL845083

Cn1cc(C(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4C(=O)c4cn(C)c5ccccc45)cc3)cc2)c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.53
CFD P00746 2/20 0.49
GFER P55789 2/20 0.48
ALDH1A1 P00352 2/20 0.48
HCRTR1 O43613 1/20 0.47
POLB P06746 1/20 0.47
CNR1 P21554 1/20 0.47
CNR2 P34972 1/20 0.47
TRPV1 Q8NER1 1/20 0.46
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 1/20 0.45
CHRM2 P08172 2/20 0.45
ADRA2A P08913 2/20 0.45
CHRM1 P11229 2/20 0.45
ADRA2B P18089 2/20 0.45
CHRM3 P20309 2/20 0.45
HTR2A P28223 2/20 0.45
HTR2C P28335 2/20 0.45
HTR4 Q13639 2/20 0.45
CYP1A2 P05177 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2195379 0.84 HSD11B1 (0.49) HSD11B1CFDGFERALDH1A1HCRTR1
SCHEMBL845332 0.84 NPC1 (0.52) CFDALDH1A1CNR1CNR2TRPV1
SCHEMBL845008 0.82 ALDH1A1 (0.54) ALDH1A1POLBCYP2C9CYP2C19CYP1A2
SCHEMBL845039 0.82 TRPV1 (0.51) ALDH1A1HCRTR1TRPV1CYP2C9CYP2C19
SCHEMBL844996 0.81 CYP2C9 (0.50) ALDH1A1TRPV1CYP2C9CYP2C19MAPK1
SCHEMBL845284 0.81 MAPK1 (0.58) ALDH1A1CYP2C9CYP2C19MAPK1HTT
SCHEMBL845131 0.80 PABPC1 (0.49) ALDH1A1TRPV1CYP2C9CYP2C19MAPK1
SCHEMBL845350 0.80 MAPK1 (0.49) ALDH1A1TRPV1CYP2C9CYP2C19CYP1A2
SCHEMBL845007 0.80 PABPC1 (0.49) ALDH1A1TRPV1CYP2C9CYP2C19MAPK1
SCHEMBL845443 0.79 CYP2C9 (0.47) ALDH1A1TRPV1CYP2C9CYP2C19MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed