SCHEMBL845095

SCHEMBL845095

CCc1cccc(C)c1C(=O)N1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)c3c(C)cccc3CC)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.47
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
CYP2C9 P11712 2/20 0.45
CYP1A2 P05177 1/20 0.45
PABPC1 P11940 1/20 0.45
CYP2C19 P33261 1/20 0.44
GAA P10253 1/20 0.43
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845333 0.94 PABPC1 (0.48) ALDH1A1MEN1KMT2ACYP2C9PABPC1
SCHEMBL845007 0.85 PABPC1 (0.49) ALDH1A1MEN1KMT2ACYP2C9PABPC1
SCHEMBL845131 0.85 PABPC1 (0.49) ALDH1A1MEN1KMT2ACYP2C9PABPC1
SCHEMBL845008 0.83 ALDH1A1 (0.54) NPSR1ALDH1A1MEN1KMT2ATDP1
SCHEMBL13272394 0.79 MEN1 (0.47) ALDH1A1MEN1KMT2ATDP1CYP2C9
SCHEMBL845697 0.79 ALDH1A1 (0.45) NPSR1ALDH1A1MEN1KMT2ATDP1
SCHEMBL845295 0.79 KDM4E (0.61) NPSR1ALDH1A1MEN1KMT2ACYP2C9
SCHEMBL845251 0.78 PABPC1 (0.50) ALDH1A1MEN1KMT2ACYP2C9PABPC1
SCHEMBL845392 0.78 ALDH1A1 (0.51) ALDH1A1MEN1KMT2ACYP2C9PABPC1
SCHEMBL845403 0.78 GFER (0.46) ALDH1A1CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed