SCHEMBL845295

SCHEMBL845295

CCOC(=O)N1CCC[C@H]1C(=O)Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)OCC)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.61
LMNA P02545 1/20 0.61
PABPC1 P11940 1/20 0.59
ALDH1A1 P00352 4/20 0.55
GAA P10253 2/20 0.55
NPC1 O15118 1/20 0.55
MAPK1 P28482 1/20 0.54
HTT P42858 1/20 0.54
HSD17B10 Q99714 1/20 0.53
NPSR1 Q6W5P4 3/20 0.52
KDM1A O60341 1/20 0.52
RCOR1 Q9UKL0 1/20 0.52
POLB P06746 1/20 0.51
TSHR P16473 3/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL872886 0.90 KDM4E (0.52) KDM4ELMNAPABPC1ALDH1A1GAA
SCHEMBL845258 0.89 MAPK1 (0.60) KDM4ELMNAPABPC1ALDH1A1NPC1
SCHEMBL844930 0.88 KDM4E (0.51) KDM4ELMNAPABPC1ALDH1A1GAA
SCHEMBL845252 0.85 KDM4E (0.73) KDM4ELMNAPABPC1ALDH1A1MAPK1
SCHEMBL844832 0.85 KDM4E (0.73) KDM4ELMNAPABPC1ALDH1A1MAPK1
SCHEMBL845251 0.85 PABPC1 (0.50) KDM4ELMNAPABPC1ALDH1A1GAA
SCHEMBL845227 0.85 NPC1 (0.76) LMNAPABPC1ALDH1A1NPC1MAPK1
SCHEMBL10299164 0.85 NPC1 (0.76) LMNAPABPC1ALDH1A1NPC1MAPK1
SCHEMBL10281278 0.85 NPC1 (0.76) LMNAPABPC1ALDH1A1NPC1MAPK1
SCHEMBL844883 0.82 KDM4E (0.69) KDM4ELMNAPABPC1ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed