SCHEMBL8451044

SCHEMBL8451044

CCc1c(C(=O)C(=O)O)c2ccccc2n1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP14 P54578 1/20 0.51
RECQL P46063 1/20 0.46
REN P00797 2/20 0.45
KDM4E B2RXH2 3/20 0.44
MAPK8 P45983 1/20 0.44
ATM Q13315 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
CYP1A2 P05177 1/20 0.44
GLA P06280 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PLA2G2A P14555 1/20 0.42
FOLH1 Q04609 1/20 0.42
PGR P06401 2/20 0.41
NR4A3 Q92570 1/20 0.41
AGTR1 P30556 3/20 0.41
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4685271 0.82 EGFR (0.49) ATML3MBTL1ALDH1A1
SCHEMBL13358189 0.79 USP14 (0.46) USP14RECQLRENKDM4EMAPK8
SCHEMBL8451877 0.77 ABCB1 (0.60) USP14RECQLKDM4EMAPK8ATM
SCHEMBL1998148 0.75 HTR6 (0.46) KDM4EATMALDH1A1HPGDCYP1A2
SCHEMBL2676368 0.72 MAPK1 (0.51) RECQLKDM4EMAPK8L3MBTL1ALDH1A1
SCHEMBL25919164 0.72 USP14 (0.55) USP14RECQLKDM4EALDH1A1HPGD
SCHEMBL1993318 0.71 CNR2 (0.55) CNR1CNR2
SCHEMBL2883770 0.71 RECQL (0.62) RECQLKDM4EALDH1A1POLBMEN1
SCHEMBL2033920 0.71 MEN1 (0.50) POLBMEN1KMT2ACNR2
SCHEMBL8702816 0.70 KMT2A (0.62) KDM4EL3MBTL1ALDH1A1HPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0624586-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-09-01 EP disclosed
US-5721230-A ANTIINFLAMMATORY AGENT, VIRICIDES; TREATING CARDIOVASCULAR DISORDER, RESPIRATORY SYSTEM DISORDER, THROMBOSIS, DIABETES, ALOPECIA HOFFMANN-LA ROCHE INC. (US) 1998-02-24 US disclosed
EP-0624586-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1994-11-17 EP disclosed