SCHEMBL4685271

SCHEMBL4685271

CCc1c(C(=O)C(=O)O)c2ccccc2n1C

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.49
OXER1 Q8TDS5 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
RAB9A P51151 1/20 0.47
ATM Q13315 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
SRC P12931 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29920927 0.83 EGFR (0.60) EGFROXER1SMN1; SMN2L3MBTL1PTGDR2
SCHEMBL8451044 0.82 USP14 (0.51) L3MBTL1ALDH1A1ATM
SCHEMBL1998148 0.80 HTR6 (0.46) EGFRALDH1A1HTTATMSRC
SCHEMBL5240303 0.79 KDM4E (0.63) SMN1; SMN2L3MBTL1ALDH1A1MAPT
SCHEMBL8702816 0.79 KMT2A (0.62) EGFRL3MBTL1ALDH1A1MAPTHTT
SCHEMBL2001294 0.77 KDM4E (0.49) ALDH1A1MAPT
SCHEMBL1993318 0.76 CNR2 (0.55)
SCHEMBL7958788 0.76 NPY1R (0.62) SMN1; SMN2L3MBTL1NPC1ALDH1A1MAPT
SCHEMBL15667319 0.76 ALDH1A1 (0.67) EGFRSMN1; SMN2L3MBTL1NPC1ALDH1A1
SCHEMBL2033920 0.76 MEN1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569901-B1 ARYL, ARYLOXY, AND ALKYLOXY SUBSTITUTED i 1H /i -INDOL-3-YL GLYOXYLIC ACID DERIVATIVES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR-1 (PAI-1) WYETH CORP (US) 2008-10-15 EP disclosed