SCHEMBL8451586

SCHEMBL8451586

N#Cc1ccc(Oc2ccncn2)cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.47
SLC22A12 Q96S37 1/20 0.41
LRRK2 Q5S007 1/20 0.39
GRIA1 P42261 2/20 0.39
GRIA2 P42262 2/20 0.39
GRIA3 P42263 2/20 0.39
GRIA4 P48058 2/20 0.39
GRM6 O15303 1/20 0.39
MAPT P10636 4/20 0.38
POLB P06746 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
APEX1 P27695 1/20 0.38
BLM P54132 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11481976 0.82 VCAM1 (0.62) VCAM1GRIA1GRIA2GRIA3GRIA4
SCHEMBL8460102 0.77 KDR (0.41) SLC22A12CYP2C9CYP19A1CYP1A2KDR
SCHEMBL8457999 0.75 CYP19A1 (0.38) SLC22A12LRRK2MAPTCYP2C9HPGD
SCHEMBL11714812 0.75 VCAM1 (0.54) VCAM1GRIA1GRIA2GRIA3GRIA4
SCHEMBL2258930 0.73 VCAM1 (0.58) VCAM1GRIA1GRIA2GRIA3GRIA4
SCHEMBL12050816 0.73 HSPB1 (0.55) MAPTPOLBALDH1A1MEN1KMT2A
SCHEMBL24750303 0.71 VCAM1 (0.49) VCAM1MAPTCYP2C9HPGDTDP1
SCHEMBL29938779 0.71 VCAM1 (0.49) VCAM1MAPTCYP2C9HPGDTDP1
SCHEMBL7689338 0.70 VCAM1 (0.54) VCAM1GRIA1GRIA2GRIA3GRIA4
SCHEMBL23887905 0.68 MAOB (0.65) VCAM1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922045-A1 BICYCLIC PYRIMIDINE DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 1999-06-16 EP disclosed
WO-1998007723-A1 BICYCLIC PYRIMIDINE DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 1998-02-26 WO disclosed