SCHEMBL8460102

SCHEMBL8460102

N#Cc1ccc(Oc2ccncn2)cc1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.41
MAPK14 Q16539 2/20 0.39
BRAF P15056 1/20 0.39
TNNI3K Q59H18 1/20 0.39
SLC22A12 Q96S37 2/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
KMO O15229 1/20 0.38
CYP19A1 P11511 2/20 0.37
PYGL P06737 1/20 0.37
PYGM P11217 1/20 0.37
XDH P47989 1/20 0.36
SCN9A Q15858 1/20 0.35
KDM4C Q9H3R0 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
PRKAB2 O43741 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20522700 0.80 KDR (0.46) KDRMAPK14BRAFTNNI3KMRGPRX4
SCHEMBL12484107 0.80 KMO (0.52) KDRMAPK14BRAFTNNI3KMRGPRX4
SCHEMBL7454153 0.79 PPARG (0.48) MRGPRX4CYP19A1PYGLPYGMCYP1A2
SCHEMBL8451586 0.77 VCAM1 (0.47) KDRMAPK14BRAFTNNI3KSLC22A12
SCHEMBL8457999 0.75 CYP19A1 (0.38) KDRMAPK14BRAFTNNI3KSLC22A12
SCHEMBL4548784 0.73 KDR (0.67) KDRMAPK14BRAFTNNI3K
SCHEMBL4309752 0.71 SMN1; SMN2 (0.54) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL11891840 0.70 SRD5A2 (0.54) KDRMAPK14BRAFTNNI3K
SCHEMBL4303621 0.68 KDR (0.42) KDRMAPK14BRAFTNNI3KKMO
SCHEMBL18906059 0.67 SRD5A2 (0.48) KDRMAPK14BRAFTNNI3KCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0922045-A1 BICYCLIC PYRIMIDINE DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 1999-06-16 EP disclosed
WO-1998007723-A1 BICYCLIC PYRIMIDINE DERIVATIVES AND THEIR USE AS ANTI-COAGULANTS SCHERING AKTIENGESELLSCHAFT (DE) 1998-02-26 WO disclosed