SCHEMBL845338

SCHEMBL845338

Cc1ccc(C(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4C(=O)c4ccc(C)nc4)cc3)cc2)cn1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RHOC P08134 1/20 0.48
RHOA P61586 1/20 0.48
NPC1 O15118 1/20 0.47
ROCK2 O75116 1/20 0.47
GRM5 P41594 3/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
PABPC1 P11940 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845297 0.85 RHOC (0.48) RHOCRHOANPC1ROCK2ALDH1A1
SCHEMBL844934 0.82 RHOC (0.51) RHOCRHOANPC1ROCK2ALDH1A1
SCHEMBL845300 0.82 CYP2C9 (0.54) RHOCRHOAROCK2ALDH1A1CYP2C9
SCHEMBL845229 0.82 RHOC (0.48) RHOCRHOANPC1ROCK2ALDH1A1
SCHEMBL845697 0.81 ALDH1A1 (0.45) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL844980 0.81 ALDH1A1 (0.45) RHOCRHOAALDH1A1CYP2C9CYP2C19
SCHEMBL844951 0.81 ROCK2 (0.55) RHOCRHOANPC1ROCK2ALDH1A1
SCHEMBL844960 0.81 DPP4 (0.43) RHOCRHOANPC1ROCK2ALDH1A1
SCHEMBL872436 0.81 DPP4 (0.43) RHOCRHOANPC1ROCK2ALDH1A1
SCHEMBL845461 0.81 PREP (0.44) RHOCRHOANPC1ROCK2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed