SCHEMBL845510

SCHEMBL845510

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3)cc2)cc1)[C@@H]1CCCN1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN3A Q9NY46 3/20 0.54
SCN9A Q15858 2/20 0.54
PSMB8 P28062 2/20 0.53
ULK1 O75385 1/20 0.49
DHODH Q02127 2/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
TERT O14746 1/20 0.46
SCN5A Q14524 1/20 0.46
JAK2 O60674 2/20 0.43
PDGFRB P09619 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL16741981 0.93 SCN3A (0.52) SCN3ASCN9APSMB8ULK1DHODH
Hydrochloric Acid SCHEMBL16741983 0.93 SCN3A (0.52) SCN3ASCN9APSMB8ULK1DHODH
SCHEMBL8236871 0.89 SCN3A (0.48) SCN3ASCN9APSMB8ULK1DHODH
SCHEMBL10119356 0.89 CA12 (0.47) SCN3ASCN9APSMB8DHODHHDAC3
SCHEMBL872523 0.88 ALDH1A1 (0.57)
SCHEMBL13388756 0.86 SCN3A (0.64) SCN3ASCN9APSMB8ULK1DHODH
SCHEMBL7692273 0.84 SCN3A (0.56) SCN3ASCN9APSMB8ULK1DHODH
SCHEMBL29365790 0.84 SCN3A (0.56) SCN3ASCN9APSMB8ULK1DHODH
SCHEMBL24609551 0.83 SCN3A (0.55) SCN3ASCN9APSMB8ULK1DHODH
SCHEMBL13379539 0.83 SCN3A (0.58) SCN3ASCN9APSMB8ULK1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed