SCHEMBL845554

SCHEMBL845554

Cn1cnc(CC(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4C(=O)c4cn(C)cn4)cc3)cc2)c1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
DGAT1 O75907 5/20 0.38
PABPC1 P11940 1/20 0.38
HCRTR1 O43613 2/20 0.38
HCRTR2 O43614 2/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
RHOC P08134 1/20 0.37
RHOA P61586 1/20 0.37
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
NPC1 O15118 1/20 0.36
MAPK1 P28482 2/20 0.36
TP53 P04637 1/20 0.36
TRHR P34981 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845391 0.94 GAA (0.42) GAAPABPC1HCRTR1HCRTR2ALDH1A1
SCHEMBL845714 0.80 HCRTR1 (0.40) GAADGAT1PABPC1HCRTR1HCRTR2
SCHEMBL844906 0.78 HCRTR1 (0.44) GAAPABPC1HCRTR1HCRTR2ALDH1A1
SCHEMBL14648097 0.77 HCRTR1 (0.42) GAAPABPC1HCRTR1HCRTR2ALDH1A1
SCHEMBL845195 0.77 HCRTR1 (0.46) GAAPABPC1HCRTR1HCRTR2ALDH1A1
SCHEMBL845393 0.75 GAA (0.47) GAAPABPC1HCRTR1HCRTR2ALDH1A1
SCHEMBL845251 0.75 PABPC1 (0.50) GAAPABPC1ALDH1A1CYP2C9CYP2C19
SCHEMBL845725 0.75 RHOC (0.45) DGAT1PABPC1ALDH1A1CYP2C9CYP2C19
SCHEMBL845620 0.74 MAPT (0.52) GAADGAT1ALDH1A1CYP2C19KDM4E
SCHEMBL845237 0.74 ALDH1A1 (0.45) GAAPABPC1HCRTR1HCRTR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed