SCHEMBL845778

SCHEMBL845778

CC(C)(C)O[C@@H]1C[C@@H](C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4C[C@@H](OC(C)(C)C)CN4C(=O)Cc4ccccc4)cc3)cc2)N(C(=O)Cc2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
HDAC8 Q9BY41 1/20 0.42
S1PR1 P21453 5/20 0.41
CYP2D6 P10635 3/20 0.41
CYP3A4 P08684 2/20 0.41
POLB P06746 1/20 0.40
CYP2C9 P11712 3/20 0.39
KMT2A Q03164 2/20 0.38
LMNA P02545 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GPR183 P32249 2/20 0.37
ALDH1A1 P00352 1/20 0.37
MMP2 P08253 2/20 0.37
ANPEP P15144 2/20 0.37
RORC P51449 1/20 0.37
KDM4E B2RXH2 1/20 0.36
BCHE P06276 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL873144 0.91 HDAC8 (0.37) CTSSCTSKHDAC8S1PR1CYP2D6
SCHEMBL845345 0.89 PAX8 (0.40) S1PR1CYP2D6CYP3A4CYP2C9KMT2A
SCHEMBL845491 0.88 POLB (0.55) POLBKMT2ALMNAMEN1NPSR1
SCHEMBL13272453 0.87 HDAC8 (0.37) CTSSCTSKHDAC8S1PR1CYP2D6
SCHEMBL845165 0.86 KDM4E (0.55) CTSKPOLBKMT2ALMNAMEN1
SCHEMBL844993 0.86 MMP2 (0.40) S1PR1CYP2D6CYP3A4CYP2C9KMT2A
SCHEMBL845768 0.85 POLB (0.49) HDAC8POLBLMNANPSR1ALDH1A1
SCHEMBL845118 0.84 POLB (0.51) POLBKMT2ALMNAMEN1NPSR1
SCHEMBL846148 0.83 POLB (0.51) CTSSCTSKHDAC8S1PR1CYP2D6
SCHEMBL845429 0.82 CTSS (0.44) CTSSCTSKHDAC8S1PR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed