SCHEMBL8457972

SCHEMBL8457972

CN(C(=O)Cc1cc(Cl)c(Cl)cc1[N+](=O)[O-])[C@@](Cc1ccccc1)(c1ccccc1)N1CCCC1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.49
OPRK1 P41145 6/20 0.40
KMT2A Q03164 1/20 0.37
OPRD1 P41143 3/20 0.35
OPRM1 P35372 2/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
UTS2R Q9UKP6 1/20 0.35
MAOA P21397 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5629630 0.71 OPRK1 (0.77) OPRK1OPRD1OPRM1ALDH1A1SMN1; SMN2
SCHEMBL8457976 0.70 OPRK1 (0.52) SIGMAR1OPRK1OPRD1OPRM1ALDH1A1
SCHEMBL5629252 0.67 SIGMAR1 (0.65) SIGMAR1OPRK1KMT2AOPRD1OPRM1
SCHEMBL6350169 0.67 SIGMAR1 (0.65) SIGMAR1OPRK1KMT2AOPRD1OPRM1
Hydrochloric Acid SCHEMBL6350294 0.66 SIGMAR1 (0.98) SIGMAR1OPRK1KMT2AOPRD1OPRM1
SCHEMBL17873685 0.65 OPRK1 (0.50) SIGMAR1OPRK1KMT2AOPRD1OPRM1
SCHEMBL5631266 0.65 OPRK1 (0.66) OPRK1OPRD1OPRM1ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL8438998 0.64 SIGMAR1 (0.41) SIGMAR1KMT2AALDH1A1SMN1; SMN2CYP1A2
SCHEMBL8433573 0.64 SIGMAR1 (0.47) SIGMAR1OPRK1KMT2ACYP2D6
SCHEMBL5630756 0.64 OPRK1 (0.63) OPRK1OPRD1OPRM1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981513-A ADMINISTERING ANTI-PRUITIC COMPOUNDS TO PATIENTS ADOLOR CORPORATION (US) 1999-11-09 US disclosed