SCHEMBL8457976

SCHEMBL8457976

CN(C(=O)Cc1cc(Cl)c(Cl)cc1[N+](=O)[O-])[C@@H](c1ccccc1)C(c1ccccc1)N1CCCC1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 14/20 0.52
SIGMAR1 Q99720 2/20 0.51
OPRD1 P41143 3/20 0.45
CYP2D6 P10635 4/20 0.43
UTS2R Q9UKP6 4/20 0.43
CYP3A4 P08684 3/20 0.43
OPRM1 P35372 2/20 0.43
TSHR P16473 2/20 0.43
CYP2C19 P33261 2/20 0.43
ALDH1A1 P00352 1/20 0.43
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5629630 0.82 OPRK1 (0.77) OPRK1OPRD1CYP2D6UTS2RCYP3A4
SCHEMBL5631266 0.75 OPRK1 (0.66) OPRK1OPRD1CYP2D6UTS2RCYP3A4
SCHEMBL5630756 0.74 OPRK1 (0.63) OPRK1OPRD1CYP2D6OPRM1
SCHEMBL8433573 0.72 SIGMAR1 (0.47) OPRK1SIGMAR1CYP2D6
SCHEMBL8457972 0.70 SIGMAR1 (0.49) OPRK1SIGMAR1OPRD1CYP2D6UTS2R
SCHEMBL5629262 0.68 OPRK1 (1.00) OPRK1SIGMAR1OPRD1CYP2D6CYP3A4
SCHEMBL8459482 0.68 OPRK1 (1.00) OPRK1SIGMAR1OPRD1CYP2D6CYP3A4
SCHEMBL5629252 0.68 SIGMAR1 (0.65) OPRK1SIGMAR1OPRD1CYP2D6CYP3A4
SCHEMBL6350169 0.68 SIGMAR1 (0.65) OPRK1SIGMAR1OPRD1CYP2D6CYP3A4
Hydrochloric Acid SCHEMBL6350294 0.67 SIGMAR1 (0.98) OPRK1SIGMAR1OPRD1CYP2D6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981513-A ADMINISTERING ANTI-PRUITIC COMPOUNDS TO PATIENTS ADOLOR CORPORATION (US) 1999-11-09 US disclosed