SCHEMBL845957

SCHEMBL845957

CNc1ccc2c(n1)CC1(C2)C(=O)Nc2ncccc21

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CALCA P06881 2/20 0.44
CALCRL Q16602 15/20 0.42
RAMP1 O60894 6/20 0.42
ADM2 Q7Z4H4 3/20 0.41
CALCB P10092 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL837518 0.85 CALCRL (0.45) CALCACALCRLRAMP1ADM2CALCB
SCHEMBL10207148 0.84 CALCA (0.46) CALCACALCRLRAMP1ADM2
SCHEMBL16658950 0.82 CALCRL (0.48) CALCACALCRLRAMP1
SCHEMBL29549672 0.82 CALCRL (0.48) CALCACALCRLRAMP1
SCHEMBL846259 0.82 CALCA (0.47) CALCACALCRLRAMP1ADM2CALCB
SCHEMBL17881436 0.82 CALCA (0.47) CALCACALCRLRAMP1ADM2CALCB
SCHEMBL837966 0.81 CALCA (0.46) CALCACALCRLRAMP1ADM2CALCB
SCHEMBL24962035 0.81 CALCRL (0.44) CALCACALCRLRAMP1
SCHEMBL877307 0.80 CALCA (0.45) CALCACALCRLRAMP1
SCHEMBL17881437 0.79 CALCRL (0.51) CALCRLRAMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143266-B2 Aryl heterocyclic CGRP receptor antagonists Merck, Sharp & Dohme Corp (US) 2012-03-27 US disclosed