Pyrrolidine

Pyrrolidine

SCHEMBL8459727

C1CCNC1.NC(O)=S.NC(O)=S.[NaH]

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
CXCR4 P61073 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NOS2 P35228 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
KMT2A Q03164 1/20 0.31
ATM Q13315 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperidine SCHEMBL10726327 0.97 ALDH1A1 (0.53) ALDH1A1CXCR4SMN1; SMN2NOS2KDM4E
Pyrrolidine SCHEMBL6853053 0.97 ALDH1A1 (0.50) ALDH1A1CXCR4SMN1; SMN2NOS2KDM4E
Pyrrolidine SCHEMBL2219944 0.97
Piperidine SCHEMBL11035777 0.94 ALDH1A1 (0.56) ALDH1A1CXCR4SMN1; SMN2NOS2KDM4E
Pyrrolidine SCHEMBL5823457 0.94 ALDH1A1 (0.47) ALDH1A1CXCR4SMN1; SMN2NOS2KDM4E
Piperidine SCHEMBL7564193 0.94 ALDH1A1 (0.56) ALDH1A1CXCR4SMN1; SMN2NOS2KDM4E
Piperidine SCHEMBL9749275 0.91 ALDH1A1 (0.53) ALDH1A1CXCR4SMN1; SMN2NOS2KDM4E
Aziridine SCHEMBL29603143 0.87
Piperidine SCHEMBL9644995 0.84 ALDH1A1 (0.60) ALDH1A1CXCR4SMN1; SMN2NOS2KDM4E
Piperazine SCHEMBL28283221 0.83 HIF1A (0.46) CXCR4SMN1; SMN2NOS2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0666741-B1 DITHIOCARBAMATES FOR THE TREATMENT OF ATHEROSCLEROSIS AND OTHER CARDIOVASCULAR AND INFLAMMATORY DISEASES UNIV EMORY (US) 1999-08-11 EP disclosed
US-5877203-A Treatment for atherosclerosis and other cardiovascular and inflammatory diseases EMORY UNIVERSITY (US) 1999-03-02 US disclosed
US-5792787-A Treatment for atherosclerosis and other cardiovascular and inflammatory diseases EMORY UNIVERSITY (US) 1998-08-11 US disclosed
EP-0666741-A1 DITHIOCARBAMATES FOR THE TREATMENT OF ATHEROSCLEROSIS AND OTHER CARDIOVASCULAR AND INFLAMMATORY DISEASES EMORY UNIVERSITY (US) 1995-08-16 EP disclosed
US-5380747-A Treatment for atherosclerosis and other cardiovascular and inflammatory diseases EMORY UNIVERSITY (US) 1995-01-10 US disclosed
WO-1994009772-A1 DITHIOCARBAMATES FOR THE TREATMENT OF ATHEROSCLEROSIS AND OTHER CARDIOVASCULAR AND INFLAMMATORY DISEASES EMORY UNIVERSITY (US) 1994-05-11 WO disclosed