SCHEMBL8463154

SCHEMBL8463154

Cc1c[c]cc(C)c1-c1cc(C(F)(F)F)c(-c2ccc(F)cc2)c(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 10/20 0.42
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
MPL P40238 1/20 0.34
PGR P06401 2/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
GABRA4 P48169 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9784280 0.83 ACHE (0.40) ARALDH1A1KDM4EGAAACHE
SCHEMBL7704882 0.79 KDM4E (0.37) ARALDH1A1KDM4EGAAMAPT
SCHEMBL7702032 0.74 AR (0.46) ARALDH1A1KDM4EGAAMAPT
SCHEMBL787753 0.72 RAPGEF4 (0.32)
SCHEMBL6941941 0.71 ACHE (0.40) ARALDH1A1ACHE
SCHEMBL27935010 0.71 AR (0.35) ARALDH1A1KMT2A
SCHEMBL26375379 0.71 NOTUM (0.46) ARALDH1A1L3MBTL1ADCY8ADCY1
SCHEMBL25844613 0.70 AR (0.49) ARALDH1A1KDM4EGAAGABRP
SCHEMBL20108386 0.66 AR (0.45) ARALDH1A1GAAMAPTKMT2A
SCHEMBL30507312 0.66 ACHE (0.48) ALDH1A1KDM4EACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906322-A1 NOVEL CHIRAL BISPHOSPHINES Merck & Co., Inc. (US) 1999-04-07 EP disclosed
WO-1997047632-A1 NOVEL CHIRAL BISPHOSPHINES MERCK & CO., INC. (US) 1997-12-18 WO disclosed