SCHEMBL8464683

SCHEMBL8464683

O=C(O)C(Cl)(Cl)CCCCCSc1cccc(-c2ccc(Cl)cc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
SHMT1 P34896 1/20 0.40
SHMT2 P34897 1/20 0.40
HDAC1 Q13547 3/20 0.40
HDAC2 Q92769 3/20 0.40
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
PTGS2 P35354 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MMP2 P08253 1/20 0.39
MEN1 O00255 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7614051 0.83 HDAC3 (0.55) KDM4EHDAC1HDAC2HDAC3HDAC4
SCHEMBL7614028 0.80 ALDH1A1 (0.53) KDM4EHDAC1HDAC2HDAC3HDAC4
SCHEMBL7619460 0.72 KDM4E (0.46) KDM4EHDAC1HDAC2HDAC3HDAC4
SCHEMBL7617774 0.72 KDM4E (0.46) KDM4EHDAC1HDAC2HDAC3HDAC4
SCHEMBL7616376 0.69 S1PR2 (0.42) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL7613532 0.69 S1PR2 (0.42) HDAC1HDAC2HDAC3HDAC4HDAC7
SCHEMBL8467642 0.69 HDAC3 (0.48) KDM4EHDAC1HDAC2HDAC3HDAC4
SCHEMBL8817718 0.69 HDAC3 (0.54) KDM4EHDAC1HDAC2HDAC3HDAC4
SCHEMBL7619484 0.68 PPARA (0.57) MEN1KMT2A
SCHEMBL682183 0.68 HDAC3 (0.49) HDAC1HDAC2HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5968982-A TREATMENT OF DIABETES ROCHE DIAGNOSTICS GMBH (DE) 1999-10-19 US disclosed