SCHEMBL8466536

SCHEMBL8466536

COc1cc(C(=O)C(=O)N(C)[C@@H](Cc2ccc(Cl)cc2)C(=O)N(C)CCC(CCC(C)c2cccnc2)c2cccnc2)cc(OC)c1OC

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CNR1 P21554 1/20 0.34
GFER P55789 1/20 0.34
LMNA P02545 2/20 0.33
ABCC1 P33527 3/20 0.33
FKBP1A P62942 1/20 0.33
FKBP4 Q02790 1/20 0.33
FKBP5 Q13451 1/20 0.33
TP53 P04637 1/20 0.33
ABCB1 P08183 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7177956 0.85 CNR1 (0.38) CYP1A2CYP2C19HSD17B10ALDH1A1CNR1
SCHEMBL7176742 0.85 CNR1 (0.38) CYP1A2CYP2C19HSD17B10ALDH1A1CNR1
SCHEMBL8463579 0.83 MAPT (0.35) ALDH1A1LMNATP53
SCHEMBL7173479 0.78 GFER (0.41) CYP1A2CYP2C19GFERLMNAFKBP1A
SCHEMBL7173487 0.78 GFER (0.41) CYP1A2CYP2C19GFERLMNAFKBP1A
SCHEMBL1492154 0.75 LPAR1 (0.39) ALDH1A1LMNAFKBP1A
SCHEMBL6472382 0.75 LPAR1 (0.39) ALDH1A1LMNAFKBP1A
SCHEMBL7181772 0.74 F10 (0.38) ALDH1A1LMNATP53
SCHEMBL7176769 0.74 F10 (0.38) ALDH1A1LMNATP53
SCHEMBL8780679 0.73 SLC2A1 (0.39) ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946190-A1 METHODS AND COMPOSITIONS FOR STIMULATING NEURITE GROWTH USING COMPOUNDS WITH AFFINITY FOR FKBP12 IN COMBINATION WITH NEUROTROPHIC FACTORS Vertex Pharmaceuticals Incorporated (US) 1999-10-06 EP claimed
WO-1998020891-A1 METHODS AND COMPOSITIONS FOR STIMULATING NEURITE GROWTH USING COMPOUNDS WITH AFFINITY FOR FKBP12 IN COMBINATION WITH NEUROTROPHIC FACTORS VERTEX PHARMACEUTICALS INCORPORATED (US) 1998-05-22 WO claimed