SCHEMBL8468665

SCHEMBL8468665

COc1nc(-c2ccncc2)sc1C=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 7/20 0.60
DBF4 Q9UBU7 7/20 0.60
CCNE1 P24864 1/20 0.60
CDK2 P24941 1/20 0.60
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
NLRP1 Q9C000 1/20 0.44
MAPT P10636 3/20 0.42
POLB P06746 1/20 0.42
HRH3 Q9Y5N1 2/20 0.42
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
PIK3CG P48736 1/20 0.40
CYP19A1 P11511 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10436914 0.84 CYP3A4 (0.49) CDC7DBF4CCNE1CDK2KDM4E
SCHEMBL27544895 0.80 CDC7 (0.49) CDC7DBF4CCNE1CDK2MEN1
SCHEMBL8705340 0.73 CDC7 (0.59) CDC7DBF4CCNE1CDK2MEN1
SCHEMBL17374890 0.72 CDC7 (0.72) CDC7DBF4CCNE1CDK2MEN1
SCHEMBL14840937 0.70 ALDH1A1 (0.38) CDC7DBF4CCNE1CDK2KMT2A
SCHEMBL8324969 0.70 CDC7 (1.00) CDC7DBF4CCNE1CDK2
SCHEMBL17374906 0.70 CDC7 (0.69) CDC7DBF4CCNE1CDK2MEN1
SCHEMBL624460 0.70 MAPT (0.44) CDC7DBF4CCNE1CDK2MEN1
SCHEMBL2517205 0.70 ALDH1A1 (0.33) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL6183091 0.70 MEN1 (0.33) MEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858444-A4 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-12-01 EP disclosed
EP-0858444-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-08-19 EP disclosed
US-5750549-A ANTIINFLAMMATORY AGENTS OR ANALGESICS MERCK & CO., INC. (US) 1998-05-12 US disclosed
WO-1997014671-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-04-24 WO disclosed