SCHEMBL8324969

SCHEMBL8324969

CCOC(=O)c1sc(-c2ccncc2)nc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 18/20 1.00
DBF4 Q9UBU7 18/20 1.00
CCNE1 P24864 1/20 0.69
CDK2 P24941 1/20 0.69
TRPM8 Q7Z2W7 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15049215 0.88 CDC7 (0.79) CDC7DBF4CCNE1CDK2TRPM8
SCHEMBL4163787 0.88 CDC7 (0.79) CDC7DBF4TRPM8
SCHEMBL5733147 0.85 CDC7 (1.00) CDC7DBF4TRPM8
SCHEMBL17374890 0.84 CDC7 (0.72) CDC7DBF4CCNE1CDK2
SCHEMBL5240574 0.84 CDC7 (1.00) CDC7DBF4TRPM8
Hydrochloric Acid SCHEMBL11121421 0.83 CDC7 (0.76) CDC7DBF4TRPM8
SCHEMBL5237288 0.81 CDC7 (0.68) CDC7DBF4TRPM8
SCHEMBL953385 0.80 CDC7 (1.00) CDC7DBF4CCNE1CDK2TRPM8
SCHEMBL17291419 0.80 CDC7 (0.70) CDC7DBF4TRPM8
SCHEMBL17374877 0.79 TRPM8 (0.75) CDC7DBF4TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858444-A4 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-12-01 EP disclosed
EP-0858444-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-08-19 EP disclosed
US-5750549-A ANTIINFLAMMATORY AGENTS OR ANALGESICS MERCK & CO., INC. (US) 1998-05-12 US disclosed
WO-1997014671-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-04-24 WO disclosed