SCHEMBL8468697

SCHEMBL8468697

O=Cc1ccc(-n2nnnc2C(F)(F)F)cn1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 2/20 0.48
HTT P42858 4/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
HPGD P15428 2/20 0.37
CACNA1B Q00975 2/20 0.37
APBA1 Q02410 2/20 0.37
HSP90AA1 P07900 1/20 0.37
CCR6 P51684 1/20 0.36
NOTUM Q6P988 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 3/20 0.32
NPSR1 Q6W5P4 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
P2RX7 Q99572 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27643287 0.79 ALDH1A1 (0.44) KCNJ1HTTALDH1A1MAPTHPGD
SCHEMBL5338473 0.74 HTT (0.40) HTTALDH1A1MAPTHPGDCACNA1B
SCHEMBL3821496 0.73 TACR1 (0.37)
SCHEMBL311546 0.72 ERN1 (0.38) HTTALDH1A1MAPTHPGDCACNA1B
SCHEMBL5432312 0.71 MEN1 (0.35) ALDH1A1
SCHEMBL310917 0.70 ALDH1A1 (0.47) HTTALDH1A1MAPTHPGDCACNA1B
SCHEMBL6100503 0.70 ALDH1A1 (0.47) HTTALDH1A1MAPTHPGDCACNA1B
SCHEMBL5551503 0.70 ALDH1A1 (0.70) HTTALDH1A1MAPTHPGDCACNA1B
SCHEMBL5549540 0.70 L3MBTL1 (0.52) HTTALDH1A1MAPTHPGDCACNA1B
SCHEMBL8464852 0.70 ALDH1A1 (0.49) HTTALDH1A1MAPTHPGDCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0858444-A4 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO INC (US) 1999-12-01 EP disclosed
EP-0858444-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 1998-08-19 EP disclosed
WO-1997014671-A1 CYCLOPENTYL TACHYKININ RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1997-04-24 WO disclosed